SCHEMBL5805979

SCHEMBL5805979

O=C1CN(c2ccccc2)c2nc(NCCc3ccc(O)cc3)ncc2N1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.56
GSK3B P49841 1/20 0.56
STAT6 P42226 7/20 0.46
ESR1 P03372 7/20 0.44
ESR2 Q92731 7/20 0.44
ULK1 O75385 1/20 0.40
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NPC1 O15118 1/20 0.36
MTOR P42345 1/20 0.36
RAB9A P51151 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
RPS6KA3 P51812 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1203451 0.73 GSK3B (0.67) GSK3AGSK3BRPS6KA3
SCHEMBL2812923 0.69 ESR2 (0.47) ESR1ESR2ADORA3ADORA2AADORA2B
SCHEMBL5805926 0.68 RPS6KA3 (0.50) STAT6ESR1ESR2ULK1RPS6KA3
SCHEMBL5816142 0.68 GSK3A (0.60) GSK3AGSK3BSTAT6ESR1ESR2
SCHEMBL1183990 0.65 KDR (0.67)
SCHEMBL1184353 0.64 KDR (0.60)
SCHEMBL10999332 0.63 HDAC3 (0.51) STAT6ADORA3ADORA2AADORA2BADORA1
Phenol SCHEMBL28213597 0.63 KDM4E (0.50) GSK3AGSK3BESR1ESR2NPC1
SCHEMBL7090103 0.62 STAT6 (0.48) GSK3AGSK3BSTAT6ESR1ESR2
SCHEMBL21502557 0.62 SCN9A (0.42) GSK3AGSK3BNPC1RAB9ARPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006091737-A1 MODULATORS OF GSK-3 ACTIVITY KEMIA, INC. (US) 2006-08-31 WO disclosed