SCHEMBL5806902

SCHEMBL5806902

CC(CO)N1CCc2cc(OCc3cccc(F)c3)ccc2C1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.55
MAOB P27338 9/20 0.47
MAOA P21397 3/20 0.47
CARM1 Q86X55 1/20 0.46
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5809330 0.89 HRH3 (0.54) HRH3MAOBMAOACARM1SLC6A2
SCHEMBL3505217 0.85 HRH3 (0.52) HRH3MAOBMAOASCN9A
SCHEMBL4430139 0.83 HRH3 (0.50) HRH3MAOBMAOASCN9A
SCHEMBL3506276 0.80 HRH3 (0.56) HRH3MAOBMAOASCN9A
SCHEMBL3506271 0.80 HRH3 (0.56) HRH3MAOBMAOASCN9A
SCHEMBL4424255 0.79 MAOB (0.60) MAOBMAOASLC6A2SLC6A4
SCHEMBL3504780 0.76 MAOB (0.56) HRH3MAOBMAOA
SCHEMBL565890 0.76 CARM1 (0.46) HRH3MAOBMAOACARM1
SCHEMBL3507700 0.75 ITGB3 (0.57) MAOBMAOACARM1
SCHEMBL5040828 0.75 MRGPRX4 (0.52) HRH3MAOBMAOASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006138475-A2 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2006-12-28 WO disclosed
EP-1501804-A1 ISOQUINOLINE DERIVATIVES MAO-B INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-02-02 EP disclosed
WO-2003091219-A1 ISOQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-06 WO disclosed