SCHEMBL5808486

SCHEMBL5808486

COc1ccc2[nH]c(C)c(CCOC(=O)NS(=O)(=O)OCCCO[N+](=O)[O-])c2c1C(=O)c1ccc(Cl)cc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.36
PTGS1 P23219 6/20 0.36
CA12 O43570 3/20 0.33
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA4 P22748 3/20 0.33
CA9 Q16790 3/20 0.33
PTGDR Q13258 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
NQO2 P16083 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
MAPT P10636 2/20 0.31
MCL1 Q07820 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5805625 0.85 PTGS2 (0.38) PTGS2PTGS1NQO2MTNR1AMTNR1B
SCHEMBL5805699 0.82 PTGS2 (0.54) PTGS2PTGS1NQO2MTNR1AMTNR1B
SCHEMBL5808398 0.81 PTGS2 (0.53) PTGS2PTGS1NQO2MTNR1AMTNR1B
SCHEMBL5805662 0.79 PTGS2 (0.38) PTGS2PTGS1CA12CA1CA2
SCHEMBL5805770 0.79 PTGS2 (0.36) PTGS2PTGS1CA12CA1CA2
SCHEMBL5809601 0.79 PTGS2 (0.55) PTGS2PTGS1CA12CA1CA2
SCHEMBL5808488 0.76 PTGS1 (0.55) PTGS2PTGS1MAPT
SCHEMBL8889810 0.75 POLB (0.39) MTNR1AMTNR1BMAPT
SCHEMBL4695816 0.75 PTGS2 (0.42) PTGS2PTGS1NQO2MTNR1AMTNR1B
SCHEMBL5808468 0.75 GAA (0.48) PTGS2PTGS1NQO2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006099416-A1 2-METHYL INDOLE CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-09-21 WO disclosed