SCHEMBL5808496

SCHEMBL5808496

Cc1c(CC(=O)NCCCO[N+](=O)[O-])c2cc(O)ccc2n1C(=O)c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 1.00
PTGS1 P23219 10/20 1.00
HRH4 Q9H3N8 1/20 0.61
CA12 O43570 1/20 0.60
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
CA4 P22748 1/20 0.60
CA9 Q16790 1/20 0.60
TRPV1 Q8NER1 1/20 0.57
HDAC3 O15379 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5806528 0.90 PTGS2 (1.00) PTGS2PTGS1HRH4CA12CA1
SCHEMBL5821337 0.86 PTGS2 (1.00) PTGS2PTGS1HRH4CA12CA1
SCHEMBL5553807 0.86 PTGS2 (0.85) PTGS2PTGS1HRH4TRPV1HDAC3
SCHEMBL5559109 0.84 PTGS2 (0.89) PTGS2PTGS1HRH4TRPV1HDAC3
SCHEMBL5555466 0.84 PTGS2 (0.82) PTGS2PTGS1HRH4TRPV1HDAC3
SCHEMBL8361039 0.82 PTGS2 (0.80) PTGS2PTGS1HRH4CA12CA1
SCHEMBL5560006 0.82 PTGS2 (0.79) PTGS2PTGS1HRH4TRPV1HDAC3
SCHEMBL5558684 0.82 PTGS2 (0.78) PTGS2PTGS1HRH4TRPV1
SCHEMBL12103292 0.81 PTGS2 (0.69) PTGS2PTGS1HRH4CA12CA1
SCHEMBL12106622 0.81 PTGS2 (0.84) PTGS2PTGS1HRH4CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006099416-A1 2-METHYL INDOLE CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-09-21 WO claimed