SCHEMBL5808917

SCHEMBL5808917

CC(=O)OOc1ccc2cc(-c3cc4ccc(C(=O)CCC(C)(C)C)cc4s3)ccc2c1Br

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.39
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
NCEH1 Q6PIU2 4/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
TNFRSF1A P19438 2/20 0.32
ALDH1A1 P00352 1/20 0.31
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5343019 0.86 PTPN1 (0.44) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL5809067 0.85 HDAC6 (0.39) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL5340323 0.83 HDAC6 (0.37) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL5337091 0.64 RXFP1 (0.46) ESR1TNFRSF1AALDH1A1PTPN1
SCHEMBL19029351 0.60 HDAC6 (0.83) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL5341289 0.60 APP (0.39) HDAC2TNFRSF1APTPN1
SCHEMBL7772381 0.59 MEN1 (0.51) NCEH1ALDH1A1
SCHEMBL16284864 0.59 SMN1; SMN2 (0.66) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL13302341 0.58 ERN1 (0.56) HDAC2ESR1ESR2
SCHEMBL8459958 0.58 HDAC6 (0.50) HDAC6HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664015-A1 SUBSTITUTED NAPHTHYL BENZOTHIOPHENE ACIDS Wyeth (US) 2006-06-07 EP disclosed
WO-2005030750-A1 SUBSTITUTED NAPHTHYL BENZOTHIOPHENE ACIDS WYETH (US) 2005-04-07 WO disclosed