SCHEMBL5809336

SCHEMBL5809336

CCOC(=O)c1cn(C2CC2)c2nc(F)c(F)cc2c1=O

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.53
DPP4 P27487 6/20 0.46
CHRM2 P08172 1/20 0.46
DRD1 P21728 1/20 0.46
KMT2A Q03164 1/20 0.46
TOP2A P11388 3/20 0.45
TOP2B Q02880 3/20 0.45
KDM4E B2RXH2 4/20 0.43
HSD17B10 Q99714 4/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
LMNA P02545 2/20 0.43
ABCC4 O15439 1/20 0.43
STAT3 P40763 1/20 0.42
MAPT P10636 1/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5422476 0.89 ADRB2 (0.51) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL10412649 0.87 ADRB2 (0.49) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL10472546 0.87 ADRB2 (0.49) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL8942057 0.86 ADRB2 (0.49) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL7230077 0.85 ADRB2 (0.50) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL10413485 0.85 ADRB2 (0.50) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL10653563 0.85 KMT2A (0.54) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL9757281 0.84 DPP4 (0.51) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL10471652 0.83 ADRB2 (0.49) ADRB2DPP4CHRM2DRD1KMT2A
SCHEMBL7005472 0.83 ADRB2 (0.49) ADRB2DPP4CHRM2DRD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed