SCHEMBL5809557

SCHEMBL5809557

COc1ccc(-c2nc(C)c3c(N)c(C(N)=O)sc3n2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.61
PIM1 P11309 4/20 0.58
KDR P35968 1/20 0.58
ABCC1 P33527 2/20 0.56
ABCG2 Q9UNQ0 2/20 0.56
IKBKB O14920 6/20 0.53
LIMK1 P53667 3/20 0.52
MAPT P10636 4/20 0.51
CDK8 P49336 2/20 0.50
CDK19 Q9BWU1 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CHUK O15111 1/20 0.50
PRKACA P17612 1/20 0.50
PRKACG P22612 1/20 0.50
PRKACB P22694 1/20 0.50
BTK Q06187 1/20 0.50
LMNA P02545 1/20 0.48
CRHBP P24387 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5805575 0.88 MAPT (0.61) ABCC1ABCG2IKBKBLIMK1MAPT
SCHEMBL6111409 0.84 IKBKB (0.64) BRAFPIM1KDRIKBKBLIMK1
SCHEMBL6112158 0.84 MAPT (0.55) IKBKBLIMK1MAPTCDK8CDK19
SCHEMBL1321257 0.83 PIM1 (0.65) BRAFPIM1KDRIKBKBLIMK1
SCHEMBL6111488 0.82 EEF2K (0.59) IKBKBLIMK1MAPTMEN1KMT2A
SCHEMBL6109707 0.82 MAPT (0.56) BRAFPIM1IKBKBLIMK1MAPT
SCHEMBL6110090 0.82 IKBKB (0.65) BRAFIKBKBLIMK1MAPTMEN1
SCHEMBL6110291 0.82 KMT2A (0.71) IKBKBLIMK1MAPTMEN1KMT2A
SCHEMBL13186380 0.81 BRAF (0.77) BRAFPIM1KDRABCC1ABCG2
SCHEMBL6110854 0.81 MAPT (0.63) IKBKBLIMK1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006100095-A1 SUBSTITUTED CARBOXAMIDES METHOD FOR PRODUCTION AND USE THEREOF AS TNF-ALPHA RELEASE INHIBITORS CURACYTE DISCOVERY GMBH (DE) 2006-09-28 WO claimed