SCHEMBL5809765

SCHEMBL5809765

Cc1cc(C2CCN(CCN(C)C(=O)O)CC2)cc(N)c1N

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.45
KDM1A O60341 1/20 0.38
SLC18A3 Q16572 2/20 0.37
OPRM1 P35372 2/20 0.36
SIGMAR1 Q99720 1/20 0.36
DRD2 P14416 3/20 0.35
DRD4 P21917 2/20 0.35
HTR7 P34969 1/20 0.35
DRD3 P35462 1/20 0.35
PLD1 Q13393 1/20 0.35
CCR5 P51681 1/20 0.34
PRCP P42785 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5805764 0.85 HRH3 (0.39) HRH3KDM1ASLC18A3OPRM1DRD2
SCHEMBL5806757 0.85 HRH3 (0.41) HRH3SIGMAR1
SCHEMBL5805753 0.72 SIGMAR1 (0.39) HRH3SIGMAR1
SCHEMBL4564154 0.72 HRH3 (0.43) HRH3KDM1ASLC18A3OPRM1DRD2
SCHEMBL5805849 0.69 HRH3 (0.45) HRH3KDM1ASLC18A3OPRM1DRD2
SCHEMBL25414060 0.67 TLR9 (0.46)
SCHEMBL14012694 0.67 HRH3 (0.47) HRH3KDM1ASLC18A3OPRM1SIGMAR1
SCHEMBL14012682 0.66 HRH3 (0.46) HRH3KDM1ASLC18A3OPRM1SIGMAR1
SCHEMBL19839243 0.66 TLR9 (0.50)
SCHEMBL16255571 0.64 SLC18A3 (0.55) SLC18A3DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006113458-A1 HETEROCYCLIC INHIBITORS OF PROTEIN ARGININE METHYL TRANSFERASES BRISTOL-MYERS SQUIBB COMPANY (US) 2006-10-26 WO disclosed