SCHEMBL581177

SCHEMBL581177

CCOC(=O)CC(=O)C1CCN(C(=O)OC)C(Cc2ccccc2C(F)(F)F)C1.COC(=O)N1CCC(C(=O)O)CC1Cc1ccccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
EPHX2 P34913 10/20 0.43
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP2C9 P11712 4/20 0.37
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HCRTR2 O43614 1/20 0.36
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP27A1 Q02318 1/20 0.35
CYP24A1 Q07973 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581437 0.96 KDM4E (0.50) KDM4EALDH1A1EPHX2SLC6A2SLC6A4
SCHEMBL3075831 0.96 KDM4E (0.50) KDM4EALDH1A1EPHX2SLC6A2SLC6A4
SCHEMBL581424 0.96 KDM4E (0.50) KDM4EALDH1A1EPHX2SLC6A2SLC6A4
SCHEMBL581930 0.90 KDM4E (0.46) KDM4EALDH1A1EPHX2CYP2C9GAA
SCHEMBL582199 0.85 ALDH1A1 (0.43) KDM4EALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL581773 0.85 ALDH1A1 (0.43) KDM4EALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL3073509 0.85 ALDH1A1 (0.43) KDM4EALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL3072810 0.82 NPSR1 (0.43) ALDH1A1GAAMEN1KMT2AL3MBTL1
SCHEMBL581342 0.82 NPSR1 (0.43) ALDH1A1GAAMEN1KMT2AL3MBTL1
SCHEMBL587229 0.82 KDM4E (0.48) KDM4EALDH1A1EPHX2CYP2C9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed