SCHEMBL5812232

SCHEMBL5812232

COc1ccc(-c2nc(N3CCN(C)CC3)sc2-c2n[c]ncc2C2CCCC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.62
ALDH1A1 P00352 5/20 0.41
CYP1A2 P05177 4/20 0.41
HSD17B10 Q99714 3/20 0.41
PTGS2 P35354 2/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 2/20 0.41
CYP2C9 P11712 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
PTGS1 P23219 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
HTR6 P50406 3/20 0.39
CETP P11597 1/20 0.38
USP2 O75604 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815362 0.99 KMT2A (0.61) KMT2AALDH1A1CYP1A2HSD17B10PTGS2
SCHEMBL5822733 0.93 KMT2A (0.51) KMT2AALDH1A1CYP1A2PTGS2TSHR
SCHEMBL5822933 0.93 KMT2A (0.51) KMT2AALDH1A1CYP1A2PTGS2TSHR
SCHEMBL5817700 0.90 KMT2A (0.48) KMT2AALDH1A1CYP1A2HSD17B10TSHR
SCHEMBL5813372 0.90 KMT2A (0.52) KMT2AALDH1A1CYP1A2HSD17B10PTGS2
SCHEMBL5819016 0.89 KMT2A (0.46) KMT2AALDH1A1CYP1A2HSD17B10CYP2C9
SCHEMBL5818863 0.87 KMT2A (0.51) KMT2AALDH1A1CYP1A2HSD17B10PTGS2
SCHEMBL5817154 0.86 KMT2A (0.50) KMT2AALDH1A1CYP1A2HSD17B10TSHR
SCHEMBL5818510 0.83 KMT2A (0.39) KMT2AALDH1A1MEN1CYP2C9KDM4E
SCHEMBL5823115 0.82 KMT2A (0.39) KMT2AALDH1A1MEN1CYP2C9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO claimed