SCHEMBL5812255

SCHEMBL5812255

Cc1c(C(C(=O)O)c2c(C)n(C(=O)c3ccc(F)c(F)c3)c3cc(F)c(O)cc23)c2cc(O)c(F)cc2n1C(=O)c1ccc(F)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
SRC P12931 1/20 0.36
PTGS2 P35354 3/20 0.35
SLC22A12 Q96S37 1/20 0.35
IGFBP3 P17936 1/20 0.34
PTGS1 P23219 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
SLC6A2 P23975 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560509 0.91 PTGS2 (0.42) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL5560592 0.91 PTGS2 (0.42) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL5550416 0.91 PTGS2 (0.42) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL5560432 0.88 AKR1C3 (0.36) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL6424980 0.88 PTGS2 (0.35) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL6424935 0.87 AKR1C3 (0.36) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL6425967 0.87 AKR1C3 (0.36) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL6425546 0.87 MEN1 (0.34) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL5560568 0.85 MEN1 (0.36) MEN1KMT2AAKR1C3AKR1C2SRC
SCHEMBL5560569 0.85 MEN1 (0.36) MEN1KMT2AAKR1C3AKR1C2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed