SCHEMBL5813077

SCHEMBL5813077

COc1ccc(CNc2nc(-c3cccnc3)nc3sc(C)c(C)c23)cc1Cl.Cc1sc2nc(-c3cccnc3)nc(Cl)c2c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
HPGD P15428 2/20 0.48
NPC1 O15118 1/20 0.48
POLB P06746 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
PDE5A O76074 3/20 0.43
MAPT P10636 2/20 0.43
PRKCI P41743 3/20 0.42
PGK1 P00558 1/20 0.41
CLK4 Q9HAZ1 3/20 0.41
DYRK1A Q13627 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
USP2 O75604 3/20 0.41
LMNA P02545 3/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
TSHR P16473 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5130031 0.97 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2HPGDNPC1POLB
SCHEMBL7174986 0.94 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2HPGDNPC1POLB
SCHEMBL7170341 0.92 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2HPGDNPC1POLB
SCHEMBL7172515 0.91 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2HPGDNPC1POLB
SCHEMBL5127640 0.90 PDE5A (0.46) ALDH1A1SMN1; SMN2HPGDNPC1POLB
SCHEMBL5130058 0.89 KMT2A (0.50) ALDH1A1SMN1; SMN2HPGDPOLBPDE5A
SCHEMBL5126022 0.87 CLK4 (0.54) ALDH1A1SMN1; SMN2HPGDNPC1POLB
SCHEMBL7016466 0.87 PDE5A (0.51) ALDH1A1SMN1; SMN2HPGDPDE5AMAPT
SCHEMBL7015902 0.87 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2HPGDPDE5AMAPT
SCHEMBL5121765 0.86 PRKCI (0.57) ALDH1A1POLBPDE5APRKCIMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed
EP-0920431-B1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2003-02-26 EP disclosed