SCHEMBL5813818

SCHEMBL5813818

CCN1C(=O)N(c2cc(OC)cc(C(=O)Nc3cc(-c4nc(C)c[nH]4)cc(C(F)(F)F)c3)c2)Cc2cnc3[nH]ccc3c21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 6/20 0.46
FGFR2 P21802 6/20 0.46
FGFR3 P22607 6/20 0.46
KDR P35968 6/20 0.46
MAP3K20 Q9NYL2 5/20 0.41
MAPK14 Q16539 5/20 0.41
ABL1 P00519 4/20 0.39
MAP4K2 Q12851 6/20 0.37
MAP3K7 O43318 5/20 0.37
TNK2 Q07912 1/20 0.37
DDR1 Q08345 1/20 0.36
NTRK1 P04629 1/20 0.36
PDGFRB P09619 1/20 0.36
KIT P10721 1/20 0.36
CSK P41240 3/20 0.36
EPHA2 P29317 2/20 0.36
MAP4K4 O95819 1/20 0.36
RAF1 P04049 1/20 0.36
LYN P07948 1/20 0.36
SRC P12931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819066 0.86 KDR (0.51) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5814241 0.84 FGFR1 (0.47) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5817693 0.82 MAP4K2 (0.50) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5819117 0.82 FGFR1 (0.47) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5819453 0.82 KDR (0.51) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5823136 0.81 FGFR1 (0.57) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5819541 0.80 KDR (0.54) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5819808 0.80 MAP3K20 (0.47) FGFR1FGFR2FGFR3KDRMAP3K20
SCHEMBL5823306 0.79 FGFR1 (0.61) FGFR1FGFR2FGFR3KDRNTRK1
SCHEMBL5819717 0.79 FGFR1 (0.61) FGFR1FGFR2FGFR3KDRNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006124731-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2006-11-23 WO disclosed