SCHEMBL5814554

SCHEMBL5814554

COc1ccc(C(C)C)cc1C(C)(C)CC(O)(Cc1[nH]c2ccccc2c1C#N)C(F)F

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 20/20 0.43
NR3C2 P08235 17/20 0.43
PGR P06401 13/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5813648 0.90 NR3C1 (0.38) NR3C1NR3C2PGR
SCHEMBL299953 0.89 NR3C1 (0.53) NR3C1NR3C2PGR
SCHEMBL5821443 0.89 NR3C1 (0.44) NR3C1NR3C2PGR
SCHEMBL5809184 0.87 NR3C1 (0.42) NR3C1NR3C2PGR
SCHEMBL27774856 0.85 NR3C1 (0.39) NR3C1NR3C2PGR
SCHEMBL5814584 0.81 NR3C1 (0.40) NR3C1NR3C2PGR
SCHEMBL13823612 0.78 NR3C1 (0.60) NR3C1NR3C2PGR
SCHEMBL291918 0.78 NR3C1 (0.46) NR3C1NR3C2PGR
SCHEMBL5781958 0.77 NR3C1 (0.51) NR3C1NR3C2PGR
SCHEMBL1634996 0.77 NR3C1 (0.68) NR3C1NR3C2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed