SCHEMBL5814799

SCHEMBL5814799

Cc1ccc(F)cc1C(C)(CC(O)(Cc1[nH]c2cnccc2c1C)C(F)(F)F)S(C)(=O)=O

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 20/20 0.79
PGR P06401 9/20 0.79
CYP3A4 P08684 4/20 0.79
NR3C2 P08235 13/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292197 0.88 NR3C1 (1.00) NR3C1PGRCYP3A4NR3C2
SCHEMBL291224 0.82 NR3C1 (0.84) NR3C1PGRCYP3A4NR3C2
SCHEMBL292871 0.82 NR3C1 (0.87) NR3C1PGRCYP3A4NR3C2
SCHEMBL5800886 0.80 NR3C1 (0.81) NR3C1PGRCYP3A4NR3C2
SCHEMBL291973 0.80 NR3C1 (0.80) NR3C1PGRCYP3A4NR3C2
SCHEMBL5797905 0.78 NR3C1 (0.77) NR3C1PGRCYP3A4NR3C2
SCHEMBL5801221 0.77 NR3C1 (0.75) NR3C1PGRCYP3A4NR3C2
SCHEMBL1932285 0.76 NR3C1 (0.74) NR3C1PGRCYP3A4NR3C2
SCHEMBL15104425 0.74 NR3C1 (0.71) NR3C1PGRCYP3A4NR3C2
SCHEMBL3689474 0.74 NR3C1 (0.65) NR3C1PGRCYP3A4NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed