SCHEMBL581875

SCHEMBL581875

COC(=O)C1CCNC(c2ccc(Cl)cc2)C1.O=C(O)C1CCN(C(=O)O)C(c2ccc(Cl)cc2)C1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SLC6A4 P31645 7/20 0.36
SLC6A3 Q01959 7/20 0.36
OPRK1 P41145 1/20 0.35
SLC6A2 P23975 6/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL581844 0.86 OPRK1 (0.36) SLC6A4SLC6A3OPRK1SLC6A2
SCHEMBL581679 0.83 SLC6A4 (0.47) SMN1; SMN2L3MBTL1SLC6A4SLC6A3SLC6A2
SCHEMBL587433 0.82 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1SLC6A4SLC6A3SLC6A2
SCHEMBL3072715 0.81 NOTUM (0.49) MEN1KMT2A
Hydrochloric Acid SCHEMBL581471 0.81 HRH3 (0.35)
Hydrochloric Acid SCHEMBL581998 0.79 MAPT (0.32)
Hydrochloric Acid SCHEMBL580915 0.78 OPRK1 (0.35) OPRK1MEN1ALDH1A1KMT2A
SCHEMBL581832 0.78 NOTUM (0.44) SMN1; SMN2L3MBTL1SLC6A4SLC6A3SLC6A2
SCHEMBL587444 0.78 SMN1; SMN2 (0.47) SMN1; SMN2L3MBTL1SLC6A4SLC6A3SLC6A2
Hydrochloric Acid SCHEMBL580918 0.76 DPP4 (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed