SCHEMBL581877

SCHEMBL581877

Cc1cc(Br)cnc1Nc1ccc(Oc2ncccc2-c2ccncc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2483671 0.81 PDE10A (0.54) PDE10A
SCHEMBL580530 0.79 PDE10A (0.53) PDE10A
SCHEMBL13282517 0.76
SCHEMBL580218 0.75 AURKA (0.56) PDE10A
SCHEMBL13282514 0.73 KCNH2 (0.57)
SCHEMBL2485954 0.73
SCHEMBL2484861 0.73
SCHEMBL13282737 0.73
SCHEMBL581766 0.72 AURKA (0.75) PDE10A
SCHEMBL2487567 0.72 PDE10A (0.54) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984353-B1 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC (US) 2015-12-30 EP disclosed
EP-2418209-B1 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC (US) 2014-06-25 EP disclosed
EP-2376455-B1 AMINOPYRIDINE AND CARBOXYPYRIDINE COMPOUNDS AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC (US) 2012-11-14 EP disclosed
EP-2418209-A1 Aurora kinase modulators and method of use Amgen Inc. (US) 2012-02-15 EP disclosed