SCHEMBL581939

SCHEMBL581939

COC(=O)c1ccnc(Cc2cccc(C(F)(F)F)c2)c1.COC(=O)c1ccnc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.51
GPR52 Q9Y2T5 5/20 0.45
NR3C2 P08235 1/20 0.44
PHGDH O43175 1/20 0.44
SCD O00767 3/20 0.43
MAOB P27338 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
MEN1 O00255 1/20 0.42
PLA2G1B P04054 1/20 0.42
GAA P10253 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ATG4B Q9Y4P1 1/20 0.42
NR1I2 O75469 1/20 0.41
ADRB1 P08588 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581494 0.94 MRGPRX4 (0.51) MRGPRX4GPR52NR3C2PHGDHSCD
SCHEMBL581445 0.81 MRGPRX4 (0.46) MRGPRX4NR3C2PHGDHMAOB
SCHEMBL581317 0.79 GPR52 (0.46) MRGPRX4GPR52CYP3A4
SCHEMBL580683 0.79 MRGPRX4 (0.55) MRGPRX4NR3C2MAOBMEN1KMT2A
SCHEMBL1568281 0.79 GPR52 (0.57) MRGPRX4GPR52NR3C2MAOB
SCHEMBL580585 0.77 KDM5B (0.56)
SCHEMBL3492157 0.76 KDM5A (0.55) MRGPRX4GPR52NR3C2PHGDH
SCHEMBL40183 0.76 MEN1 (0.68) MRGPRX4CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL7776064 0.75 HTR2B (0.46) GPR52MAOBCYP1A2CYP3A4CYP2D6
SCHEMBL31750237 0.75 HTR2B (0.46) GPR52MAOBCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed