SCHEMBL5819944

SCHEMBL5819944

CNc1cccc(-c2ccnc3c(C(=O)c4ccccc4)cnn23)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 4/20 0.57
MAPK13 O15264 2/20 0.57
MAP2K1 Q02750 1/20 0.56
CLK4 Q9HAZ1 1/20 0.56
DYRK1B Q9Y463 1/20 0.56
TLR8 Q9NR97 1/20 0.55
BRAF P15056 7/20 0.55
GSK3A P49840 3/20 0.55
EPHA2 P29317 1/20 0.55
CDKN1A P38936 1/20 0.54
LIMK1 P53667 2/20 0.53
MARK2 Q7KZI7 1/20 0.53
AKT1 P31749 1/20 0.53
PIM3 Q86V86 1/20 0.53
MAPK9 P45984 1/20 0.51
DYRK1A Q13627 1/20 0.51
IRAK4 Q9NWZ3 1/20 0.51
KDM4E B2RXH2 1/20 0.50
CDK1 P06493 1/20 0.50
MAPKAPK2 P49137 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361381 0.91 PIM1 (0.60) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL10733510 0.90 GSK3A (0.59) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL7361513 0.90 MAPK13 (0.54) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL10731559 0.89 MAP2K1 (0.53) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL5823296 0.88 BRAF (0.57) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL7363602 0.88 MAPK13 (0.57) PIM1MAPK13BRAFGSK3AEPHA2
SCHEMBL7362738 0.86 CLK4 (0.73) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL5816204 0.85 PIM1 (0.59) PIM1MAPK13BRAFGSK3AEPHA2
SCHEMBL5822141 0.85 CDKN1A (0.75) PIM1MAPK13MAP2K1CLK4DYRK1B
SCHEMBL5819755 0.85 CDKN1A (0.74) PIM1MAPK13MAP2K1CLK4DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006033795-A2 SUBSTITUTED PYRAZOLO [1, 5-A] PYRIMIDINES FOR INHIBITING ABNORMAL CELL GROWTH WYETH (US) 2006-03-30 WO disclosed
US-4654347-A USEFUL AS ANXIOLYTIC AND ANTIEPILEPTIC AGENTS, SEDATIVE-HYPNOTIC AGENTS AND SKELETAL MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1987-03-31 US disclosed