SCHEMBL5819954

SCHEMBL5819954

O=C(NC1CCC(C(=O)O)CC1)c1cc(F)cnc1Cl

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.49
DGAT1 O75907 5/20 0.44
JAK2 O60674 2/20 0.42
NTRK1 P04629 2/20 0.42
CRHR1 P34998 3/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
P2RX7 Q99572 1/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4D Q08499 1/20 0.41
MCHR1 Q99705 1/20 0.39
MAP4K4 O95819 2/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8353042 0.87 HPGD (0.51) HPGDJAK2CRHR1RAB9ANPC1
SCHEMBL5778940 0.87 HPGD (0.51) HPGDJAK2NTRK1CRHR1RAB9A
SCHEMBL5778937 0.87 HPGD (0.51) HPGDJAK2NTRK1CRHR1RAB9A
SCHEMBL8349012 0.86 HPGD (0.46) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL6063963 0.86 HPGD (0.46) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL8352231 0.86 HPGD (0.50) HPGDJAK2CRHR1RAB9ANPC1
SCHEMBL5841319 0.86 SMYD3 (0.52) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL5841315 0.86 SMYD3 (0.52) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL3174715 0.85 NPC1 (0.58) HPGDRAB9ANPC1SMN1; SMN2GAA
Hydrochloric Acid SCHEMBL6063550 0.85 SMYD3 (0.51) HPGDCRHR1RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651609-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS Pfizer Limited (GB) 2006-05-03 EP disclosed
WO-2005009966-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed