SCHEMBL8353042

SCHEMBL8353042

O=C(N[C@H]1CC[C@@H](NCl)CC1)c1cc(F)cnc1Cl

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.51
CRHR1 P34998 5/20 0.44
RAB9A P51151 3/20 0.44
NPC1 O15118 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4D Q08499 1/20 0.42
MAP4K4 O95819 2/20 0.41
MCHR1 Q99705 1/20 0.41
P2RX7 Q99572 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
POLB P06746 1/20 0.39
SMYD3 Q9H7B4 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778937 0.89 HPGD (0.51) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL5778940 0.89 HPGD (0.51) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL8352231 0.88 HPGD (0.50) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL5841319 0.88 SMYD3 (0.52) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL5841315 0.88 SMYD3 (0.52) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL3174715 0.88 NPC1 (0.58) HPGDRAB9ANPC1SMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL6063550 0.87 SMYD3 (0.51) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL5819954 0.87 HPGD (0.49) HPGDCRHR1RAB9ANPC1SMN1; SMN2
SCHEMBL8296522 0.86 HPGD (0.48) HPGDRAB9ANPC1SMN1; SMN2SMYD3
SCHEMBL6063963 0.84 HPGD (0.46) HPGDCRHR1RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003068233-A1 NICOTINAMIDE DERIVATIVES AND A TIOTROPIUM SALT IN COMBINATION FOR THE TREATMENT OF E.G. INFLAMMATORY, ALLERGIC AND RESPIRATORY DISEASES PFIZER LIMITED (GB) 2003-08-21 WO disclosed