SCHEMBL5820046

SCHEMBL5820046

CC1(C)OCC(CC(C)(C)c2cc(Br)cc3c2OCC3)(C(F)F)O1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.39
PGR P06401 1/20 0.39
NR3C2 P08235 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4490217 0.82 NR3C1 (0.42) NR3C1PGRNR3C2
Dimethylamine SCHEMBL5822669 0.81 NR3C1 (0.35) NR3C1PGRNR3C2
SCHEMBL5822670 0.80 NR3C1 (0.33) NR3C1PGRNR3C2
SCHEMBL5363258 0.77 NR3C1 (0.46) NR3C1PGRNR3C2
SCHEMBL5363254 0.77 NR3C1 (0.46) NR3C1PGRNR3C2
SCHEMBL5814888 0.70 NR3C1 (0.46) NR3C1PGRNR3C2
SCHEMBL820526 0.68 PTGS1 (0.46) NR3C1PGRNR3C2
SCHEMBL4489826 0.68 NR3C1 (0.30) NR3C1PGRNR3C2
SCHEMBL1633800 0.66 NR3C1 (0.48) NR3C1PGRNR3C2
SCHEMBL15756223 0.66 NR3C1 (0.37) NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed