SCHEMBL5820537

SCHEMBL5820537

[c]1nnc(-c2ncco2)o1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.34
LTA4H P09960 1/20 0.33
ADRA2A P08913 2/20 0.31
ADRA1A P35348 2/20 0.31
ADRA1D P25100 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL100765 0.76 HPGDS (0.46) HPGDSLTA4HADRA2AADRA1AADRA1D
SCHEMBL9455041 0.68 HPGDS (0.35) HPGDSLTA4H
SCHEMBL16799432 0.68 NOTUM (0.42)
SCHEMBL569960 0.65 NPC1 (0.48)
SCHEMBL9454206 0.65 HPGDS (0.37) HPGDSLTA4H
SCHEMBL5820538 0.65 NOTUM (0.43) HPGDS
SCHEMBL967548 0.64 PDPK1 (0.38)
SCHEMBL4032194 0.64 KDM4E (0.48)
SCHEMBL5200683 0.64 HPGDS (0.35) HPGDSLTA4H
SCHEMBL17701202 0.63 HPGDS (0.35) HPGDSLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658069-A1 HETEROCYCLIC AMIDE DERIVATIVES WHICH POSSESS GLYCOGEN PHOSPHORYLASE INHIBITORY ACTIVITY Astrazeneca AB (SE) 2006-05-24 EP disclosed
WO-2005013981-A1 HETEROCYCLIC AMIDE DERIVATIVES WHICH POSSESS GLYCOGEN PHOSPHORYLASE INHIBITORY ACTIVITY ASTRAZENECA AB (SE) 2005-02-17 WO disclosed