SCHEMBL582069

SCHEMBL582069

CCOC(=O)CC(=O)C1CCN(C(=O)OC)C(c2ccc(C(F)(F)F)c(F)c2)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(C(F)(F)F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.42
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 2/20 0.35
NOTUM Q6P988 2/20 0.35
KDM1A O60341 1/20 0.34
TRPM8 Q7Z2W7 2/20 0.33
ANXA2 P07355 1/20 0.33
S100A10 P60903 1/20 0.33
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581628 0.97 EPHX2 (0.44) EPHX2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL580803 0.89 NOTUM (0.42) EPHX2NOTUMKDM1ATRPM8
SCHEMBL581321 0.89 EPHX2 (0.37) EPHX2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL581320 0.89 EPHX2 (0.37) EPHX2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL3080499 0.89 EPHX2 (0.37) EPHX2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL581727 0.87 NOTUM (0.38) ALDH1A1KDM4ENOTUMTDP1
SCHEMBL581726 0.87 NOTUM (0.38) ALDH1A1KDM4ENOTUMTDP1
SCHEMBL3072590 0.86 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1
SCHEMBL3072798 0.86 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1
SCHEMBL580838 0.86 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed