SCHEMBL582159

SCHEMBL582159

COC(=O)C1CCNC(Cc2cc(F)cc(F)c2)C1.O=C(O)C1CCN(C(=O)O)C(Cc2cc(F)cc(F)c2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.36
ALDH1A1 P00352 3/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
BACE1 P56817 2/20 0.31
MMP1 P03956 2/20 0.31
ADAM17 P78536 2/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
ABCB1 P08183 1/20 0.31
TACR1 P25103 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
PLG P00747 1/20 0.30
DPP4 P27487 1/20 0.30
DPP8 Q6V1X1 1/20 0.30
DPP9 Q86TI2 1/20 0.30
DPP7 Q9UHL4 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581020 0.87 OPRK1 (0.35) OPRK1ALDH1A1MAPTHPGDNPSR1
SCHEMBL580821 0.84 PLG (0.38) BACE1PLGDPP4DPP8DPP9
SCHEMBL580937 0.84 TACR1 (0.41) ALDH1A1MAPTHPGDNPSR1HSD17B10
SCHEMBL587768 0.83 NOTUM (0.37) OPRK1TACR1
SCHEMBL587405 0.80 OPRK1 (0.43) OPRK1ALDH1A1MAPTHPGDNPSR1
SCHEMBL581731 0.80 PSEN1 (0.36) OPRK1ALDH1A1MAPTHPGDNPSR1
SCHEMBL581126 0.75 MAPT (0.40) ALDH1A1MAPTTACR1PLGHTT
SCHEMBL580826 0.74 PLG (0.50) MMP1ADAM17PLG
SCHEMBL580910 0.74 TACR1 (0.45) TACR1
SCHEMBL586999 0.74 OPRK1 (0.35) OPRK1ALDH1A1MAPTHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed