SCHEMBL5821909

SCHEMBL5821909

CC(C)(C)[SiH2]OC(C)(C)c1cccc2[nH]c(-c3nn(Br)c4ncccc34)nc12

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.33
CBFB Q13951 4/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
AURKA O14965 2/20 0.31
CXCR3 P49682 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821904 0.75 CDK1 (0.42) CDK1CBFBALDH1A1TP53CYP3A4
SCHEMBL4040032 0.71 RET (0.43) CDK1AURKA
SCHEMBL5465608 0.60 NOS3 (0.40) SMN1; SMN2
SCHEMBL124272 0.56 CBFB (0.68) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL21237321 0.55 PKN1 (0.57) ALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL14738396 0.55 CHEK1 (0.30)
SCHEMBL1585571 0.54 ELANE (0.49) ALDH1A1HPGDHSD17B10
SCHEMBL22599976 0.53 MGAM (0.48) CBFB
SCHEMBL3443410 0.53 ELANE (0.36) ALDH1A1TP53HPGDSMN1; SMN2
SCHEMBL5455968 0.52 METAP1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006130673-A1 3-BENZOIMIDAZOLYL-PYRAZOLOPYRIDINES USEFUL IN TREATING KINASE DISORDERS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-12-07 WO disclosed