SCHEMBL5822896

SCHEMBL5822896

COc1ccc(-n2c(CN3CCC[C@H]3C(=O)O)nnc2-c2ccc(-c3cccc(C)c3C)cn2)cn1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OXTR P30559 6/20 0.53
AVPR1A P37288 6/20 0.53
AVPR2 P30518 2/20 0.53
CD274 Q9NZQ7 14/20 0.46
PDCD1 Q15116 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931120 0.93 OXTR (0.52) OXTRAVPR1AAVPR2CD274PDCD1
SCHEMBL931030 0.84 OXTR (0.61) OXTRAVPR1AAVPR2CD274
SCHEMBL930550 0.80 OXTR (0.80) OXTRAVPR1AAVPR2
SCHEMBL930956 0.78 OXTR (0.41) OXTRAVPR1AAVPR2
SCHEMBL5121875 0.74 OXTR (0.60) OXTRAVPR1AAVPR2
SCHEMBL6532411 0.73 OXTR (0.69) OXTRAVPR1AAVPR2
SCHEMBL931377 0.73 OXTR (0.80) OXTRAVPR1AAVPR2
SCHEMBL931016 0.70 OXTR (0.69) OXTRAVPR1AAVPR2
SCHEMBL8279842 0.70 OXTR (0.42) OXTRAVPR1AAVPR2
SCHEMBL930950 0.70 OXTR (1.00) OXTRAVPR1AAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673355-A1 SUBSTITUTED TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS Pfizer Limited (GB) 2006-06-28 EP disclosed
WO-2005028452-A1 SUBSTITUTED TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-03-31 WO disclosed