SCHEMBL582398

SCHEMBL582398

CN1CCC(=O)CC1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A5 Q9Y345 1/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
CHKA P35790 1/20 0.36
HDAC1 Q13547 1/20 0.36
P2RX7 Q99572 1/20 0.36
PLCG1 P19174 1/20 0.36
AADAT Q8N5Z0 1/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5850350 0.81 ABCB1 (0.41) HRH3
Iodide SCHEMBL28776545 0.80 ABCB1 (0.40) HRH3
SCHEMBL3076567 0.79 KMT2A (0.44) KDM4EP2RX7KCNH2HRH3
SCHEMBL27852924 0.78 AKR1B10 (0.37) TACR1KDM4EALDH1A1KCNH2HRH3
SCHEMBL12056397 0.77 KDM4E (0.43) KDM4EALDH1A1CHKACARM1PRMT6
SCHEMBL7684256 0.75 TACR1 (0.55) TACR1ALDH1A1
SCHEMBL12266683 0.72 TEAD1 (0.43) SLC6A2SLC6A4HCRTR1HCRTR2P2RX7
SCHEMBL13963553 0.70
SCHEMBL4991727 0.69 HTR2C (0.39) SLC6A2SLC6A4P2RX7
SCHEMBL19411415 0.69 ABCB1 (0.36) TACR1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed