SCHEMBL5828716

SCHEMBL5828716

CCc1c(-c2ccccc2)c2c(c3c1[nH]c1ccc(O)cc13)C(=O)NC2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 14/20 1.00
WEE1 P30291 13/20 1.00
ROCK2 O75116 4/20 0.65
GSK3A P49840 1/20 0.63
GSK3B P49841 1/20 0.63
CDK5 Q00535 1/20 0.63
CDK5R1 Q15078 1/20 0.63
MEN1 O00255 1/20 0.60
PRKD3 O94806 1/20 0.60
PRKCG P05129 1/20 0.60
PRKCB P05771 1/20 0.60
CDK4 P11802 1/20 0.60
PRKCA P17252 1/20 0.60
PRKCH P24723 1/20 0.60
PRKCI P41743 1/20 0.60
PRKCE Q02156 1/20 0.60
KMT2A Q03164 1/20 0.60
PRKCQ Q04759 1/20 0.60
PRKCZ Q05513 1/20 0.60
PRKCD Q05655 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5829135 0.88 CHEK1 (1.00) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL5829403 0.86 CHEK1 (1.00) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL5829223 0.85 CHEK1 (1.00) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL5828138 0.84 CHEK1 (0.73) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL8120620 0.80 ROCK2 (1.00) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL5829194 0.78 CHEK1 (1.00) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL27047988 0.77 CHEK1 (0.74) CHEK1WEE1ROCK2GSK3AGSK3B
SCHEMBL6516584 0.75 WEE1 (1.00) CHEK1WEE1MEN1PRKD3PRKCG
SCHEMBL29414147 0.75 WEE1 (1.00) CHEK1WEE1MEN1PRKD3PRKCG
SCHEMBL30250020 0.75 WEE1 (1.00) CHEK1WEE1MEN1PRKD3PRKCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed