SCHEMBL5830574

SCHEMBL5830574

Cc1c(Cc2cccc(C(F)(F)F)c2F)c2ccc(Cl)c(Cl)c2n1CCCNS(C)(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 3/20 0.36
P2RX7 Q99572 8/20 0.35
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32
GRIA2 P42262 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
RECQL P46063 1/20 0.30
CYSLTR2 Q9NS75 1/20 0.30
CYSLTR1 Q9Y271 1/20 0.30
CD38 P28907 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5673140 0.81 TRPV4 (0.40) TRPV4POLBL3MBTL1HTR2AHTR2C
SCHEMBL5675120 0.75 TDP1 (0.39) TRPV4LMNARECQLRORC
SCHEMBL476597 0.71 CNR2 (0.46) TRPV4P2RX7RORC
SCHEMBL5934979 0.71 TRPV4 (0.38) TRPV4LMNACD38HTR2AHTR2C
SCHEMBL5831060 0.71 TRPV4 (0.36) TRPV4P2RX7POLBL3MBTL1CD38
SCHEMBL5656870 0.70 KMT2A (0.40) TRPV4POLB
SCHEMBL6228793 0.69 TRPV4 (0.33) TRPV4POLBL3MBTL1
SCHEMBL6230901 0.69 TRPV4 (0.35) TRPV4
SCHEMBL476632 0.68 CNR2 (0.46) TRPV4
SCHEMBL476653 0.66 CNR2 (0.47) TRPV4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7138424-B2 Indole derivatives, method for preparing same and pharmaceutical compositions containing same SANOFI-AVENTIS (FR) 2006-11-21 US disclosed
US-20060089345-A1 Indole derivatives, method for preparating same and pharmaceutical compositions containing same SANOFI-AVENTIS (FR) 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089345-A1 Indole derivatives, method for preparating same and pharmaceutical compositions containing same CNR2, CNR1, IDO2 TRPV4 208/4885P2RX7 84/4885POLB 4798/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.