SCHEMBL5833165

SCHEMBL5833165

O=Cc1cc2ccnc(-c3ccc(Cl)cc3)c2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.45
TDO2 P48775 2/20 0.45
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
MAPK13 O15264 6/20 0.38
MAPK12 P53778 6/20 0.38
MAPK11 Q15759 6/20 0.38
MAPK14 Q16539 6/20 0.38
GCGR P47871 5/20 0.38
MAPT P10636 1/20 0.36
RAF1 P04049 1/20 0.35
CYP2A6 P11509 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
SCN9A Q15858 1/20 0.34
CCNB2 O95067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4275395 0.80 CYP2A6 (0.42) MAPTCYP2A6
SCHEMBL1735901 0.78 IDO1 (0.48) IDO1TDO2PDE3BPDE3AMAPK13
SCHEMBL24896318 0.69 CYP2A6 (0.38) MAPTCYP2A6
SCHEMBL14484408 0.66 PDE3B (0.41) IDO1TDO2PDE3BPDE3AMAPK13
SCHEMBL20853236 0.66 TNF (0.44) MAPTCYP2A6
SCHEMBL20840621 0.65 DAO (0.53) MAPTCYP2A6KDM4E
SCHEMBL26912475 0.65 CYP2A6 (0.43) MAPTCYP2A6
SCHEMBL20571353 0.64 ALDH1A1 (0.42) MAPTCYP2A6KDM4E
SCHEMBL19154063 0.64 TRIM24 (0.47) IDO1TDO2PDE3BPDE3AMAPT
SCHEMBL12284018 0.64 SCN2A (0.51) MAPTKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732566-A2 6-AZAINDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2006-12-20 EP disclosed
WO-2005097129-A2 6-AZAINDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-10-20 WO disclosed