Bicarbonate

Bicarbonate

SCHEMBL583862

CCn1nc(C)c2c(NC3CCCCC3)c(C3=NOC4(CCC(C(=O)NC)CC4)C3)cnc21.O=C(O)O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
PDE4B Q07343 9/20 0.37
PDE7A Q13946 2/20 0.37
KMT2A Q03164 2/20 0.31
NR3C1 P04150 2/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL582947 0.93 POLB (0.45) POLBPDE4BPDE7AKMT2ANR3C1
SCHEMBL582686 0.93 POLB (0.47) POLBPDE4BPDE7AKMT2APDE3B
Bicarbonate SCHEMBL582961 0.93 POLB (0.46) POLBPDE4BPDE7AKMT2ANR3C1
SCHEMBL582541 0.92 POLB (0.48) POLBPDE4BPDE7AKMT2ANR3C1
Bicarbonate SCHEMBL583229 0.92 POLB (0.46) POLBPDE4BPDE7AKMT2ANR3C1
SCHEMBL582381 0.92 POLB (0.47) POLBPDE4BPDE7AKMT2ANR3C1
Bicarbonate SCHEMBL583789 0.91 POLB (0.50) POLBPDE4BPDE7AKMT2ANR3C1
Bicarbonate SCHEMBL583188 0.91 POLB (0.50) POLBPDE4BPDE7AKMT2ANR3C1
Bicarbonate SCHEMBL583374 0.91 POLB (0.50) POLBPDE4BPDE7AKMT2ANR3C1
SCHEMBL583157 0.91 POLB (0.44) POLBPDE4BPDE7AKMT2APDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124944-B1 Pyrazolo[3,4-b]pyridine derivatives as phosphodiesterase inhibitors RANBAXY LAB LTD (IN) 2012-02-15 EP claimed