SCHEMBL5839079

SCHEMBL5839079

CC(C)n1cnc2c(Nc3ccc([N+](=O)[O-])cc3)nc(Cl)nc21

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 10/20 0.68
CDK5R1 Q15078 10/20 0.68
CDK2 P24941 10/20 0.68
CCNA2 P20248 9/20 0.68
CCNA1 P78396 9/20 0.68
DYRK1A Q13627 8/20 0.68
NPC1 O15118 1/20 0.68
POLB P06746 1/20 0.68
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
CCNE2 O96020 1/20 0.53
CCNE1 P24864 1/20 0.53
CDK1 P06493 4/20 0.52
ADORA2A P29274 1/20 0.48
FLT3 P36888 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4489273 0.87 CDK5 (0.66) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL183351 0.85 MEN1 (0.61) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL5839686 0.82 CDK5 (0.76) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL28771433 0.82 CDK2 (0.76) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL6574754 0.82 ADORA2A (0.58) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL5827777 0.82 CDK5 (0.79) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL23494096 0.81 CDK5 (1.00) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL31307877 0.81 CDK5 (1.00) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL17212875 0.79 CDK5 (0.78) CDK5CDK5R1CDK2CCNA2CCNA1
SCHEMBL17212872 0.78 CDK5 (1.00) CDK5CDK5R1CDK2CCNA2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed
CN-1066147-C Purine derivatives and process for preparing same 诺瓦提斯公司 2001-05-23 CN disclosed
CN-1202896-A Purine derivatives and processes for their preparation 诺瓦提斯公司 1998-12-23 CN disclosed
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed