SCHEMBL5839709

SCHEMBL5839709

COc1cccc(Nc2nc(Cl)nc3c2ncn3C(C)C)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 12/20 0.69
CDK5R1 Q15078 12/20 0.69
CCNA2 P20248 10/20 0.69
CDK2 P24941 10/20 0.69
CCNA1 P78396 10/20 0.69
DYRK1A Q13627 9/20 0.67
NPC1 O15118 1/20 0.58
POLB P06746 1/20 0.58
CDK1 P06493 7/20 0.55
CCNB1 P14635 3/20 0.55
CCNB2 O95067 2/20 0.55
CCNB3 Q8WWL7 2/20 0.55
KDM4E B2RXH2 2/20 0.55
MAPK1 P28482 2/20 0.55
EIF2AK2 P19525 1/20 0.54
GSK3B P49841 1/20 0.54
MERTK Q12866 1/20 0.54
MEN1 O00255 1/20 0.52
PAK4 O96013 1/20 0.52
CCNE2 O96020 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5840458 0.86 CDK5 (0.74) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL29444630 0.86 CDK5 (0.74) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL20549706 0.85 CDK5 (0.73) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL5839477 0.84 CDK5 (0.72) CDK5CDK5R1CCNA2CDK2CCNA1
Hydrochloric Acid SCHEMBL5840186 0.84 CDK1 (0.55) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL5827777 0.84 CDK5 (0.79) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL5839410 0.83 CDK1 (0.69) CDK5CDK5R1CCNA2CDK2NPC1
SCHEMBL1443458 0.82 CDK1 (0.80) CDK5CCNA2CDK2CCNA1NPC1
SCHEMBL17212873 0.82 CDK5 (1.00) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL5840389 0.81 CDK1 (0.75) CDK5CDK5R1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed