SCHEMBL5840147

SCHEMBL5840147

CCn1cnc2c(Nc3cccc(Cl)c3)nc(NC(CO)CO)nc21

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 14/20 0.74
MAPT P10636 4/20 0.72
KDM4E B2RXH2 3/20 0.72
NPC1 O15118 3/20 0.72
CDK5 Q00535 3/20 0.72
CDK5R1 Q15078 3/20 0.72
POLB P06746 1/20 0.72
PRKCA P17252 5/20 0.68
NPSR1 Q6W5P4 1/20 0.68
TDP1 Q9NUW8 1/20 0.68
CCNB1 P14635 5/20 0.62
TP53 P04637 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP3A4 P08684 2/20 0.62
CYP2D6 P10635 2/20 0.62
CDK4 P11802 2/20 0.62
TSHR P16473 2/20 0.62
CCNA2 P20248 2/20 0.62
CCND1 P24385 2/20 0.62
CCNE1 P24864 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8706894 0.96 CDK5 (0.78) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL8710243 0.96 CDK5 (0.78) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5841668 0.96 CDK5 (0.78) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5840882 0.89 CDK1 (0.72) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5840894 0.89 CDK1 (0.72) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5839355 0.85 CDK1 (1.00) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5840472 0.85 CDK1 (0.67) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5841742 0.85 CDK1 (0.72) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5841752 0.85 CDK1 (0.72) CDK1MAPTKDM4ENPC1CDK5
SCHEMBL5840718 0.83 CDK1 (0.73) CDK1MAPTKDM4ENPC1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed