SCHEMBL8710243

SCHEMBL8710243

CC[C@@H](CO)Nc1nc(Nc2cccc(Cl)c2)c2ncn(CC)c2n1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.78
MAPT P10636 4/20 0.78
CDK5R1 Q15078 4/20 0.78
KDM4E B2RXH2 3/20 0.78
NPC1 O15118 3/20 0.78
POLB P06746 1/20 0.78
CDK1 P06493 14/20 0.72
NPSR1 Q6W5P4 1/20 0.66
TDP1 Q9NUW8 1/20 0.66
PRKCA P17252 5/20 0.66
CCNB1 P14635 5/20 0.61
CCNA2 P20248 3/20 0.61
CCNE1 P24864 3/20 0.61
CDK2 P24941 3/20 0.61
TP53 P04637 2/20 0.61
CYP1A2 P05177 2/20 0.61
CYP3A4 P08684 2/20 0.61
CYP2D6 P10635 2/20 0.61
CDK4 P11802 2/20 0.61
TSHR P16473 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5841668 1.00 CDK5 (0.78) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL8706894 1.00 CDK5 (0.78) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5840147 0.96 CDK1 (0.74) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5840882 0.91 CDK1 (0.72) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5840894 0.91 CDK1 (0.72) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5841752 0.89 CDK1 (0.72) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5841742 0.89 CDK1 (0.72) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5839851 0.87 CDK1 (0.67) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL7208712 0.87 CDK1 (0.73) CDK5MAPTCDK5R1KDM4ENPC1
SCHEMBL5839860 0.87 CDK1 (0.67) CDK5MAPTCDK5R1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed