SCHEMBL5840706

SCHEMBL5840706

CCn1cnc2c(Nc3cccc(C#N)c3)nc(Cl)nc21

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 15/20 0.69
PRKCA P17252 6/20 0.69
NPC1 O15118 2/20 0.68
YTHDC1 Q96MU7 1/20 0.63
CTSV O60911 1/20 0.53
CTSL P07711 1/20 0.53
CTSB P07858 1/20 0.53
CTSH P09668 1/20 0.53
CTSS P25774 1/20 0.53
CTSK P43235 1/20 0.53
CASP4 P49662 1/20 0.53
MMP14 P50281 1/20 0.53
CTSC P53634 1/20 0.53
BACE1 P56817 1/20 0.53
ADAM17 P78536 1/20 0.53
CTSZ Q9UBR2 1/20 0.53
KLK4 Q9Y5K2 1/20 0.53
CCNB1 P14635 2/20 0.49
CLK1 P49759 2/20 0.49
CLK2 P49760 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3352454 0.85 NPC1 (0.74) CDK1PRKCANPC1YTHDC1CCNB1
SCHEMBL29444624 0.85 NPC1 (0.74) CDK1PRKCANPC1YTHDC1CCNB1
SCHEMBL5840317 0.84 CDK1 (0.68) CDK1PRKCANPC1CTSVCTSL
SCHEMBL3379300 0.83 YTHDC1 (0.60) CDK1PRKCANPC1YTHDC1CCNA2
SCHEMBL5840449 0.82 CDK1 (1.00) CDK1PRKCANPC1
SCHEMBL5839910 0.82 CDK1 (0.69) CDK1PRKCANPC1CCNB1CLK1
SCHEMBL5839410 0.82 CDK1 (0.69) CDK1PRKCANPC1YTHDC1CCNB1
Hydrochloric Acid SCHEMBL5839390 0.81 CDK1 (1.00) CDK1PRKCANPC1
SCHEMBL3346901 0.81 NPC1 (1.00) CDK1PRKCANPC1CTSVCTSL
SCHEMBL5839344 0.80 CDK1 (0.68) CDK1PRKCANPC1CCNB1CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed