SCHEMBL5845398

SCHEMBL5845398

CC(O)Cn1ncc2ccc(O)c([N+](=O)[O-])c21

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 14/20 0.49
HTR2C P28335 14/20 0.49
HTR2B P41595 7/20 0.49
MAPK1 P28482 1/20 0.42
ATM Q13315 1/20 0.42
LMNA P02545 1/20 0.42
HTR1A P08908 2/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
HTR1D P28221 1/20 0.36
HTR7 P34969 1/20 0.36
HTR4 Q13639 1/20 0.36
CHRM1 P11229 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
KMO O15229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5845389 1.00 HTR2A (0.49) HTR2AHTR2CHTR2BMAPK1ATM
SCHEMBL5638272 0.83 HTR2A (0.46) HTR2AHTR2CHTR2BMAPK1ATM
SCHEMBL5638269 0.83 HTR2A (0.46) HTR2AHTR2CHTR2BMAPK1ATM
SCHEMBL5845487 0.83 HTR2A (0.46) HTR2AHTR2CHTR2BMAPK1ATM
SCHEMBL5843691 0.77 HTR2C (0.55) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL5845010 0.77 HTR2C (0.58) HTR2AHTR2CHTR2BLMNAHTR1A
SCHEMBL5843697 0.77 HTR2C (0.55) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL5845013 0.77 HTR2C (0.58) HTR2AHTR2CHTR2BLMNAHTR1A
SCHEMBL27140224 0.76 ESR1 (0.39) HTR2AHTR2CHTR2BESR1ESR2
SCHEMBL5844513 0.76 HTR2C (0.51) HTR2AHTR2CHTR2BHTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7129257-B1 Pyrazolo[3,4- e]benzoxazoles for the treatment of glaucoma ALCON, INC. (CH) 2006-10-31 US disclosed