SCHEMBL5846277

SCHEMBL5846277

COC(=O)COc1ccc(C(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 15/20 1.00
CXCR2 P25025 15/20 1.00
P4HTM Q9NXG6 1/20 0.55
GABRA5 P31644 1/20 0.54
ALDH1A1 P00352 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
ATM Q13315 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5846984 0.94 CXCR1 (1.00) CXCR1CXCR2P4HTMNPC1RAB9A
SCHEMBL5847552 0.89 CXCR1 (0.80) CXCR1CXCR2P4HTMGABRA5ALDH1A1
SCHEMBL5846287 0.89 CXCR1 (1.00) CXCR1CXCR2P4HTMGABRA5ALDH1A1
SCHEMBL5846063 0.88 CXCR1 (0.79) CXCR1CXCR2P4HTMGABRA5ALDH1A1
SCHEMBL5847588 0.87 CXCR1 (0.83) CXCR1CXCR2GABRA5
SCHEMBL5846254 0.87 CXCR2 (0.78) CXCR1CXCR2P4HTMGABRA5
SCHEMBL5845966 0.85 CXCR1 (0.80) CXCR1CXCR2
SCHEMBL5845511 0.85 CXCR2 (1.00) CXCR1CXCR2P4HTMGABRA5
SCHEMBL5658349 0.85 CXCR2 (0.73) CXCR1CXCR2P4HTMALDH1A1NPC1
SCHEMBL5847596 0.84 CXCR1 (1.00) CXCR1CXCR2P4HTMGABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6777432-B1 TREATING A SUBJECT HAVING AN INFLAMMATORY DISORDER ALLEVIATED BY THE INHIBITION OF GRO- ALPHA CYTOKINES DARWIN MOLECULAR CORPORATION 2004-08-17 US claimed
US-7151112-B1 Pharmaceutical uses and synthesis of nicotinamides UCB SA (GB) 2006-12-19 US disclosed
US-6777432-B1 TREATING A SUBJECT HAVING AN INFLAMMATORY DISORDER ALLEVIATED BY THE INHIBITION OF GRO- ALPHA CYTOKINES DARWIN MOLECULAR CORPORATION 2004-08-17 US disclosed