SCHEMBL5658349

SCHEMBL5658349

COC(=O)COc1ncc(C(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 15/20 0.73
CXCR1 P25024 14/20 0.73
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
ATM Q13315 1/20 0.52
P4HTM Q9NXG6 1/20 0.51
ALDH1A1 P00352 1/20 0.50
PTPN1 P18031 1/20 0.48
PTPN6 P29350 1/20 0.48
PTPN11 Q06124 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5656391 0.89 CXCR1 (0.75) CXCR2CXCR1P4HTMALDH1A1
SCHEMBL5659069 0.89 CXCR2 (0.59) CXCR2CXCR1NPC1RAB9AATM
SCHEMBL5659634 0.88 CXCR1 (0.58) CXCR2CXCR1NPC1RAB9AATM
SCHEMBL5661096 0.87 CXCR2 (0.67) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL5656328 0.86 P4HTM (0.57) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL5846277 0.85 CXCR1 (1.00) CXCR2CXCR1NPC1RAB9AATM
SCHEMBL5656795 0.84 CXCR2 (0.76) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL5660344 0.84 CXCR1 (0.57) CXCR2CXCR1P4HTMALDH1A1
SCHEMBL5660642 0.83 CXCR2 (0.75) CXCR2CXCR1P4HTM
SCHEMBL5658045 0.83 CXCR2 (0.59) CXCR2CXCR1NPC1RAB9AP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed