SCHEMBL5846774

SCHEMBL5846774

COC(=O)[C@H]1Cc2cc(S(=O)(=O)Cl)ccc2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 3/20 0.40
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
RECQL P46063 1/20 0.39
SCN3A Q9NY46 1/20 0.38
GABRA1 P14867 1/20 0.37
GABRB2 P47870 1/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
TBXA2R P21731 1/20 0.36
CYP2D6 P10635 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
OPRK1 P41145 1/20 0.36
MTNR1A P48039 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5846780 1.00 GLS (0.40) GLSPOLBAPEX1RECQLSCN3A
SCHEMBL5846771 1.00 GLS (0.40) GLSPOLBAPEX1RECQLSCN3A
SCHEMBL5848095 0.87 CYP4F2 (0.48) POLBMEN1KMT2ACYP2D6OPRK1
SCHEMBL5848090 0.87 CYP4F2 (0.48) POLBMEN1KMT2ACYP2D6OPRK1
SCHEMBL5848089 0.87 CYP4F2 (0.48) POLBMEN1KMT2ACYP2D6OPRK1
SCHEMBL5848677 0.82 GLA (0.47) MEN1KMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL5848676 0.82 GLA (0.47) MEN1KMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL5848675 0.82 GLA (0.47) MEN1KMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL4455342 0.81 GLS (0.56) GLSPOLBGABRA1GABRB2MEN1
SCHEMBL29443014 0.81 GLS (0.56) GLSPOLBGABRA1GABRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7034051-B2 Fused bicyclic carboxamide derivatives and methods of their use ADOLOR CORPORATION (US) 2006-04-25 US disclosed
US-20050054630-A1 Fused bicyclic carboxamide derivatives and methods of their use CUBIST PHARMACEUTICALS, INC. 2005-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054630-A1 Fused bicyclic carboxamide derivatives and methods of their use PAICS, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CPS1 GLS 14/4885POLB 852/4885APEX1 4308/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.