SCHEMBL5847185

SCHEMBL5847185

COc1ccc(-c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CC3)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
ALDH1A1 P00352 2/20 0.39
STS P08842 2/20 0.39
CCR3 P51677 2/20 0.39
HTT P42858 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GPR119 Q8TDV5 3/20 0.38
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848624 1.00 HTR2A (0.44) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5847743 0.94 HTR2A (0.48) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5847917 0.92 HTR2A (0.46) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5847114 0.91 HTR2A (0.45) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5847234 0.91 CNR1 (0.41) ALDH1A1STSMEN1KMT2AGPR119
SCHEMBL5847616 0.90 HTR2A (0.46) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5847319 0.89 HTR2A (0.44) HTR2AHTR2CHTR2BALDH1A1STS
SCHEMBL5413294 0.89 HTR2C (0.46) HTR2AHTR2CHTR2BCCR3MEN1
SCHEMBL5420008 0.89 HTR2C (0.46) HTR2AHTR2CHTR2BCCR3MEN1
SCHEMBL5847795 0.89 HTR2A (0.59) HTR2AHTR2CHTR2BALDH1A1STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed