SCHEMBL5847795

SCHEMBL5847795

COc1ccc(-c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CC3)c(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.59
HTR2C P28335 1/20 0.59
HTR2B P41595 1/20 0.59
EPHX2 P34913 2/20 0.47
GPR119 Q8TDV5 3/20 0.39
ALDH1A1 P00352 2/20 0.38
STS P08842 2/20 0.38
CCR3 P51677 2/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
PROKR1 Q8TCW9 3/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SRC P12931 2/20 0.36
ABL1 P00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848217 0.95 HTR2A (0.66) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5416044 0.95 HTR2A (0.66) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5847212 0.94 HTR2A (0.63) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5848068 0.93 HTR2A (0.65) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5847472 0.92 HTR2A (0.49) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5847300 0.91 HTR2A (0.49) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5847616 0.90 HTR2A (0.46) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5847917 0.90 HTR2A (0.46) HTR2AHTR2CHTR2BEPHX2GPR119
SCHEMBL5408675 0.90 HTR2A (0.62) HTR2AHTR2CHTR2BEPHX2CCR3
SCHEMBL6503159 0.90 HTR2A (0.51) HTR2AHTR2CHTR2BEPHX2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed