SCHEMBL5847313

SCHEMBL5847313

COc1ccc(-c2cc3c4c(c2)[C@@H]2CN(C(=O)OC(C)(C)C)CC[C@@H]2N4CCC3)c(C)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51
GPR119 Q8TDV5 3/20 0.40
ALDH1A1 P00352 3/20 0.39
STS P08842 2/20 0.39
PIK3CA P42336 2/20 0.38
PRKDC P78527 2/20 0.38
MTOR P42345 1/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
TSHR P16473 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SRC P12931 2/20 0.37
PDE4B Q07343 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848103 0.98 HTR2A (0.49) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5847114 0.95 HTR2A (0.45) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5848188 0.90 HTR2A (0.50) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5847291 0.90 HTR2A (0.49) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5416044 0.90 HTR2A (0.66) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5848217 0.90 HTR2A (0.66) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5405383 0.89 HTR2C (0.53) HTR2AHTR2CHTR2BALDH1A1MEN1
SCHEMBL5847431 0.89 HTR2A (0.50) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5847743 0.89 HTR2A (0.48) HTR2AHTR2CHTR2BGPR119ALDH1A1
SCHEMBL5848505 0.89 HTR2A (0.48) HTR2AHTR2CHTR2BGPR119ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed