SCHEMBL584822

SCHEMBL584822

CC(C)(C)OC(=O)N1CC[C@@H](O)C[C@H]1C(C)(C)O[SiH2]C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
HSD17B10 Q99714 1/20 0.34
PREP P48147 1/20 0.34
HPGD P15428 1/20 0.33
RECQL P46063 1/20 0.32
EPHX1 P07099 1/20 0.32
USP2 O75604 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL585463 1.00 CHRM2 (0.41) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL4274094 0.86 CHRM2 (0.40) CHRM2CHRM1CHRM3HSD17B10CYP1A2
SCHEMBL3243618 0.86 CHRM2 (0.40) CHRM2CHRM1CHRM3HSD17B10CYP1A2
SCHEMBL18660256 0.82 CHRM2 (0.49) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL15058137 0.79 CHRM2 (0.46) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL21073336 0.79 CHRM2 (0.46) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL15058138 0.79 CHRM2 (0.46) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL21073334 0.79 CHRM2 (0.46) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL15058136 0.79 CHRM2 (0.46) CHRM2CHRM1CHRM3HSD17B10PREP
SCHEMBL3248189 0.77 NR1H2 (0.34) CHRM2CHRM1CHRM3CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102217-B1 4- (2-OXO-OXAZOLIDIN-3YL)-PHENOXYMETHYLE DERIVATIVEAS AS ANTIBACTERIALS ACTELION PHARMACEUTICALS LTD (CH) 2012-02-15 EP disclosed
US-8039466-B2 5-hydroxymethyl-oxazolidin-2-one antibacterials ACTELION PHARMACEUTICAL LTD. (CH) 2011-10-18 US disclosed
US-20100069376-A1 5-HYDROXYMETHYL-OXAZOLIDIN-2-ONE ANTIBACTERIALS ACTELION PHARMACEUTICALS, LTD. (CH) 2010-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069376-A1 5-HYDROXYMETHYL-OXAZOLIDIN-2-ONE ANTIBACTERIALS OGFOD1, ODC1, OXGR1 CHRM2 1192/4885CHRM1 365/4885CHRM3 1048/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.