SCHEMBL5848258

SCHEMBL5848258

CC(C)(C)OC(=O)N1CC[C@H]2[C@@H](C1)c1cc(-c3ccc(Cl)c(Cl)c3)cc3c1N2CCCC3

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
OPRK1 P41145 1/20 0.39
KAT6A Q92794 1/20 0.38
KAT5 Q92993 1/20 0.38
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPN6 P29350 1/20 0.38
USP30 Q70CQ3 2/20 0.37
GPR119 Q8TDV5 2/20 0.37
NTRK1 P04629 1/20 0.37
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
HTR2A P28223 3/20 0.35
HTR2C P28335 3/20 0.35
DRD2 P14416 2/20 0.35
HTR2B P41595 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5846974 0.97 NPC1 (0.40) NPC1RAB9AOPRK1KAT6AKAT5
SCHEMBL5849606 0.94 PTPN2 (0.39) NPC1RAB9AOPRK1KAT6AKAT5
SCHEMBL5848083 0.91 USP30 (0.40) NPC1RAB9APTPN2PTPN1PTPN6
SCHEMBL5847512 0.89 STS (0.41) NPC1RAB9AKAT6AKAT5USP30
SCHEMBL5847125 0.89 TP53 (0.42) NPC1RAB9AKAT6AKAT5USP30
SCHEMBL5847308 0.89 USP30 (0.41) NPC1RAB9APTPN2PTPN1PTPN6
SCHEMBL5847676 0.88 GPR119 (0.39) NPC1RAB9AUSP30GPR119CNR1
SCHEMBL5849542 0.88 STS (0.40) NPC1RAB9AUSP30HTR2AHTR2C
SCHEMBL5847077 0.88 NPC1 (0.40) NPC1RAB9APTPN2PTPN1PTPN6
SCHEMBL5847225 0.87 MEN1 (0.39) NPC1RAB9AUSP30GPR119PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed