SCHEMBL5848583

SCHEMBL5848583

NC(=O)C1CCCCc2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.46
EPHX1 P07099 1/20 0.46
IDO1 P14902 2/20 0.45
HTT P42858 1/20 0.44
MCL1 Q07820 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ANO1 Q5XXA6 1/20 0.43
F2 P00734 1/20 0.43
F12 P00748 1/20 0.43
CRBN Q96SW2 4/20 0.42
BLM P54132 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3812210 0.95 IDO1 (0.50) PIN1EPHX1IDO1HTTALDH1A1
SCHEMBL29934643 0.95 IDO1 (0.50) PIN1EPHX1IDO1HTTALDH1A1
SCHEMBL177082 0.95 IDO1 (0.50) PIN1EPHX1IDO1HTTALDH1A1
SCHEMBL5732694 0.95 IDO1 (0.50) PIN1EPHX1IDO1HTTALDH1A1
SCHEMBL30252198 0.95 IDO1 (0.50) PIN1EPHX1IDO1HTTALDH1A1
Bromide SCHEMBL3727457 0.93 IDO1 (0.49) PIN1EPHX1IDO1HTTALDH1A1
Hydrochloric Acid SCHEMBL3726157 0.93 IDO1 (0.51) PIN1EPHX1IDO1HTTALDH1A1
SCHEMBL2475968 0.87 PIN1 (0.58) PIN1IDO1CRBN
SCHEMBL29528570 0.87 PIN1 (0.58) PIN1IDO1CRBN
SCHEMBL643577 0.87 PIN1 (0.58) PIN1IDO1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7034051-B2 Fused bicyclic carboxamide derivatives and methods of their use ADOLOR CORPORATION (US) 2006-04-25 US disclosed
WO-2005023799-A1 FUSED BICYCLIC CARBOXAMIDE DERIVATIVES AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2005-03-17 WO disclosed
US-20050054630-A1 Fused bicyclic carboxamide derivatives and methods of their use CUBIST PHARMACEUTICALS, INC. 2005-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054630-A1 Fused bicyclic carboxamide derivatives and methods of their use PAICS, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CPS1 PIN1 2503/4885EPHX1 2789/4885IDO1 2514/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.