SCHEMBL5851682

SCHEMBL5851682

Cc1cc2c(N3CCN(C(=O)OC(C)(C)C)CC3)ncnc2s1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.55
P2RY12 Q9H244 6/20 0.49
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
MEN1 O00255 5/20 0.47
KMT2A Q03164 1/20 0.45
HTT P42858 2/20 0.44
LMNA P02545 1/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
MAP4K4 O95819 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
GBA1 P04062 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5851315 0.88 KIT (0.54) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5850542 0.88 KIT (0.54) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5848798 0.88 KIT (0.57) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5849579 0.87 KIT (0.53) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5851715 0.86 MAPT (0.57) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5850552 0.86 P2RY12 (0.68) P2RY12ALDH1A1KDM4ESMN1; SMN2MAPT
SCHEMBL5849376 0.85 KIT (0.52) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5849530 0.85 KIT (0.52) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5849427 0.84 P2RY12 (0.57) KITP2RY12ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5849216 0.84 P2RY12 (0.55) KITP2RY12ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115741-B2 4-thieno[2,3-D]pyrimidin-4-YL piperazine compounds ALEXION PHARMACEUTICALS, INC. 2006-10-03 US disclosed
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed