SCHEMBL5860841

SCHEMBL5860841

COc1ccc(C(C)(CC(=O)O)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.47
ITGA4 P13612 1/20 0.47
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
ALOX15 P16050 1/20 0.44
APEX1 P27695 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 1/20 0.42
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 1/20 0.40
EPHX2 P34913 1/20 0.40
KMT2A Q03164 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31477659 0.85 CYP2C19 (0.54) MAPK1RECQLTDP1NPC1RAB9A
SCHEMBL1573515 0.85 CYP2C19 (0.54) MAPK1RECQLTDP1NPC1RAB9A
SCHEMBL5862223 0.85 CYP2C19 (0.54) MAPK1RECQLTDP1NPC1RAB9A
SCHEMBL5862815 0.84 MIF (0.49) ITGB1ITGA4ALDH1A1MAPTPPARG
SCHEMBL6513375 0.84 HIF1A (0.39) ITGB1ITGA4MAPK1RECQLTDP1
SCHEMBL7971106 0.83 CXCR2 (0.40) ITGB1ITGA4PPARGPPARACA1
SCHEMBL6517072 0.80 ALDH1A1 (0.48) ALDH1A1LMNAMAPK1RECQLMAPT
SCHEMBL27159467 0.78 MAPT (0.45) ALDH1A1LMNAALOX15APEX1MAPK1
SCHEMBL27159469 0.78 MAPT (0.45) ALDH1A1LMNAALOX15APEX1MAPK1
SCHEMBL12834968 0.77 MAPT (0.46) ALDH1A1LMNAALOX15APEX1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7041667-B1 CCR5 modulators PFIZER, INC. (US) 2006-05-09 US disclosed
EP-1013276-A1 Aminoazacycloalkanes as CCR5 modulators PFIZER INC. (US) 2000-06-28 EP disclosed