SCHEMBL5860855

SCHEMBL5860855

NC(=O)N(c1ccc(Oc2ccccc2)cc1)c1ccc2cn(CCCN3CCC[C@H]3CO)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
MCHR1 Q99705 4/20 0.41
MCHR2 Q969V1 2/20 0.41
FGFR3 P22607 3/20 0.37
KDR P35968 3/20 0.37
FGFR1 P11362 2/20 0.37
FGFR2 P21802 2/20 0.37
FGFR4 P22455 2/20 0.37
BTK Q06187 4/20 0.37
LTA4H P09960 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
TERT O14746 1/20 0.36
SCN9A Q15858 2/20 0.35
SPHK1 Q9NYA1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5860521 0.86 MCHR1 (0.42) ALDH1A1MCHR1MCHR2BTK
SCHEMBL5862064 0.82 MCHR1 (0.58) ALDH1A1MCHR1MCHR2TERT
SCHEMBL5862261 0.81 MCHR1 (0.45) ALDH1A1MCHR1SCN9A
SCHEMBL6348132 0.79 MCHR1 (0.45) ALDH1A1MCHR1MCHR2BTK
SCHEMBL5860936 0.77 MCHR1 (0.41) ALDH1A1MCHR1BTK
SCHEMBL6374843 0.75 NPSR1 (0.45) ALDH1A1MCHR1FGFR3KDRFGFR1
SCHEMBL5860935 0.75 MCHR1 (0.69) MCHR1MCHR2
SCHEMBL5861989 0.74 MCHR1 (0.57) MCHR1MCHR2TERT
SCHEMBL6380408 0.74 MCHR1 (0.64) ALDH1A1MCHR1MCHR2LTA4HHRH3
SCHEMBL5861302 0.73 MCHR1 (0.58) MCHR1MCHR2TERT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049307-B2 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor ABBOTT LABORATORIES (US) 2006-05-23 US claimed
US-20050187279-A1 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor ABBVIE INC. 2005-08-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050187279-A1 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor MCHR1, MCHR2, MC1R ALDH1A1 2303/4885MCHR1 1/4885MCHR2 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.